Kinase Inhibitors AGC Akt-I-1 AKT Serine-Threonine 473382-39-7 NU1005-001 1 mg 195.00 NU1005-005 5 mg 385.00 NU1005-010 10 mg 605.00 NU1005-050 50 mg 1,750.00 Akt-I-2 AKT Serine-Threonine 473382-48-8 NU1006-001 1 mg 195.00 NU1006-005 5 mg 385.00 NU1006-010 10 mg 605.00 NU1006-050 50 mg 1,750.00 BI-D1870 S6K Serine-Threonine 501437-28-1 NU1020-001 1 mg 90.00 NU1020-005 5 mg 170.00 NU1020-010 10 mg 265.00 NU1020-050 50 mg 655.00 Bisindoylmaleimide X PKC, PLCbeta Serine-Threonine 145317-11-9 NU1021-001 1 mg 125.00 (Ro 31-8425) NU1021-005 5 mg 210.00 NU1021-010 10 mg 310.00 NU1021-050 50 mg 870.00 BX795 PDK1 Serine-Threonine 702675-74-9 NU1026-001 1 mg 65.00 NU1026-005 5 mg 100.00 NU1026-010 10 mg 135.00 NU1026-050 50 mg 540.00 BX912 PDK1, PI3K Serine-Threonine 702674-56-4 NU1027-001 1 mg 65.00 NU1027-005 5 mg 140.00 NU1027-010 10 mg 220.00 NU1027-050 50 mg 640.00 GSK-690693 AKT Serine-Threonine 937174-76-0 NU1043-001 1 mg 70.00 NU1043-005 5 mg 120.00 NU1043-010 10 mg 165.00 NU1043-050 50 mg 755.00 GSK429286A ROCK Serine-Threonine 864082-47-3 NU1071-001 1 mg 90.00 (RHO-15) NU1071-005 5 mg 155.00 NU1071-010 10 mg 230.00 NU1071-050 50 mg 665.00 SR3677 RSK Serine-Threonine 1072959-67-1 NU1083-001 1 mg 100.00 NU1083-005 5 mg 155.00 NU1083-010 10 mg 210.00 NU1083-050 50 mg 760.00 A-674563 AKT, PKA, CDK7, Serine-Threonine 552325-73-2 NU1110-001 1 mg 175.00 CDK5, CDK4, CDK2 NU1110-005 5 mg 270.00 NU1110-010 10 mg 450.00 NU1110-050 50 mg 1,490.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 1
Merck-22-6 AKT Serine-Threonine 12847-42-4 NU1118-001 1 mg 385.00 NU1118-005 5 mg 650.00 NU1118-010 10 mg 945.00 NU1118-050 50 mg 2,740.00 GSK-25 RSK1, p70s6k Serine-Threonine 874119-56-9 NU1124-001 1 mg 190.00 NU1124-005 5 mg 385.00 NU1124-010 10 mg 605.00 NU1124-050 50 mg 1,925.00 R428 AKT Serine-Threonine 1037624-75-1 NU1131-001 1 mg 250.00 NU1131-005 5 mg 650.00 NU1131-010 10 mg 1,200.00 NU1131-050 50 mg 3,900.00 S6K-18 S6K Serine-Threonine 1265789-88-5 NU1132-001 1 mg 190.00 NU1132-005 5 mg 385.00 NU1132-010 10 mg 540.00 NU1132-050 50 mg 1,485.00 AZD-26 AKT Serine-Threonine 1357158-81-6 NU1160-001 1 mg 195.00 NU1160-005 5 mg 385.00 NU1160-010 10 mg 605.00 NU1160-050 50 mg 1,750.00 MK-2206 AKT Serine-Threonine 1032350-13-2 NU1162-001 1 mg 70.00 (MK-2206 dihydrochloride) NU1162-005 5 mg 110.00 NU1162-010 10 mg 170.00 NU1162-050 50 mg 555.00 Ruboxistaurin PKC Serine-Threonine 169939-93-9 NU1172-001 1 mg 165.00 (LY333531) NU1172-005 5 mg 275.00 NU1172-010 10 mg 430.00 NU1172-050 50 mg 1,310.00 PF-04708671 S6K1 Serine-Threonine 1255517-76-0 NU1177-001 1 mg 60.00 NU1177-005 5 mg 140.00 NU1177-010 10 mg 205.00 NU1177-050 50 mg 800.00 Atypical (PIKK) Selumetinib mtor Serine-Threonine 606143-52-6 NU1016-001 1 mg 80.00 (AZD6244, ARRY142886) NU1016-005 5 mg 120.00 NU1016-010 10 mg 200.00 NU1016-050 50 mg 590.00 BEZ-235 mtor, PI3K Serine-Threonine 915019-65-7 NU1018-001 1 mg 60.00 (NVP-BEZ235) NU1018-005 5 mg 90.00 NU1018-010 10 mg 130.00 NU1018-050 50 mg 165.00 KU0063794 mtor Serine-Threonine 938440-64-3 NU1050-001 1 mg 70.00 NU1050-005 5 mg 90.00 NU1050-010 10 mg 150.00 NU1050-050 50 mg 450.00 KU55933 ATM/ATR Serine-Threonine 587871-26-9 NU1051-001 1 mg 50.00 NU1051-005 5 mg 70.00 NU1051-010 10 mg 120.00 NU1051-050 50 mg 360.00 AMG-51 mtor Serine-Threonine 890019-63-3 NU1111-001 1 mg 190.00 NU1111-005 5 mg 385.00 NU1111-010 10 mg 605.00 NU1111-050 50 mg 1,815.00 AMG-458 mtor Serine-Threonine 913376-83-7 NU1144-001 1 mg 125.00 NU1144-005 5 mg 260.00 NU1144-010 10 mg 355.00 NU1144-050 50 mg 1,050.00 AZD8055 mtor Serine-Threonine 1009298-09-2 NU1166-001 1 mg 60.00 (CCG 168) NU1166-005 5 mg 100.00 NU1166-010 10 mg 115.00 NU1166-050 50 mg 320.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 2
AZD2014 mtor Serine-Threonine 1009298-59-2 NU1167-001 1 mg 100.00 NU1167-005 5 mg 150.00 NU1167-010 10 mg 250.00 NU1167-050 50 mg 980.00 IPI 145 mtor, PI3K Serine-Threonine 1201438-56-3 NU1175-001 1 mg 105.00 NU1175-005 5 mg 165.00 NU1175-010 10 mg 275.00 NU1175-050 50 mg 930.00 Rapamycin mtor Serine-Threonine 53123-88-9 NU1185-001 1 mg 50.00 (Sirolimus, AY-22989, NU1185-005 5 mg 70.00 WY-090217) NU1185-010 10 mg 100.00 NU1185-050 50 mg 385.00 CAMK AZD7762 Chk1 Serine-Threonine 860352-01-8 NU1017-001 1 mg 80.00 NU1017-005 5 mg 100.00 NU1017-010 10 mg 160.00 NU1017-050 50 mg 490.00 CX-4945 Chk2 Serine-Threonine 1009820-21-6 NU1109-001 1 mg 100.00 NU1109-005 5 mg 165.00 NU1109-010 10 mg 275.00 NU1109-050 50 mg 825.00 SMI-4a PIM Serine-Threonine 438190-29-5 NU1113-001 1 mg 50.00 NU1113-005 5 mg 75.00 NU1113-010 10 mg 130.00 NU1113-050 50 mg 320.00 SCH 900776 Chk1, Chk2 Serine-Threonine 891494-63-6 NU1173-001 1 mg 105.00 NU1173-005 5 mg 210.00 NU1173-010 10 mg 370.00 NU1173-050 50 mg 950.00 PF0477736 Chk1 Serine-Threonine 952021-60-2 NU1174-001 1 mg 65.00 NU1174-005 5 mg 145.00 NU1174-010 10 mg 210.00 NU1174-050 50 mg 645.00 XL388 Chk1 Serine-Threonine 1251156-08-7 NU1186-001 1 mg 155.00 NU1186-005 5 mg 265.00 NU1186-010 10 mg 360.00 NU1186-050 50 mg 1,265.00 SGI-1776 Pim1, Pim2, Pim3 Serine-Threonine 1025065-69-3 NU1193-001 1 mg 80.00 NU1193-005 5 mg 130.00 NU1193-010 10 mg 220.00 NU1193-050 50 mg 715.00 CMGC AT-7519 CDK2, CDK7, Serine-Threonine 902135-91-5 NU1010-001 1 mg 60.00 CDK5, CDK4 NU1010-005 5 mg 100.00 NU1010-010 10 mg 150.00 NU1010-050 50 mg 540.00 CC-401 JNK Serine-Threonine 395104-30-0 NU1028-001 1 mg 115.00 NU1028-005 5 mg 200.00 NU1028-010 10 mg 310.00 NU1028-050 50 mg 1,045.00 Alvocidib CDK2, CDK7, Serine-Threonine 146426-40-6 NU1040-001 1 mg 60.00 (Flavopiridol, HMR-1275, CDK4, CDK5 NU1040-005 5 mg 100.00 L868275) NU1040-010 10 mg 130.00 NU1040-050 50 mg 385.00 Purvalanol B CDK2, CDK7, Serine-Threonine 212844-54-7 NU1070-001 1 mg 50.00 (NG95) CDK5, CDK4 NU1070-005 5 mg 75.00 NU1070-010 10 mg 100.00 NU1070-050 50 mg 385.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 3
RWJ-67657 p38 Serine-Threonine 215303-72-3 NU1072-001 1 mg 50.00 NU1072-005 5 mg 75.00 NU1072-010 10 mg 100.00 NU1072-050 50 mg 385.00 SB202190 p38 Serine-Threonine 152121-30-7 NU1073-001 1 mg 50.00 NU1073-005 5 mg 65.00 NU1073-010 10 mg 95.00 NU1073-050 50 mg 260.00 SB202190 HCl p38 Serine-Threonine 350228-36-3 NU1073A-001 1 mg 50.00 NU1073A-005 5 mg 65.00 NU1073A-010 10 mg 95.00 NU1073A-050 50 mg 260.00 SB203580 p38 Serine-Threonine 152121-47-6 NU1074-001 1 mg 50.00 (RWJ 64809, PB 203580) NU1074-005 5 mg 65.00 NU1074-010 10 mg 75.00 NU1074-050 50 mg 220.00 SB-242235 p38 Serine-Threonine 193746-75-7 NU1076-001 1 mg 190.00 NU1076-005 5 mg 385.00 NU1076-010 10 mg 605.00 NU1076-050 50 mg 1,815.00 SD-06 p38 Serine-Threonine 271576-80-8 NU1078-001 1 mg 190.00 NU1078-005 5 mg 385.00 NU1078-010 10 mg 605.00 NU1078-050 50 mg 1,815.00 SD169 MAPK, p38 Serine-Threonine 1670-87-7 NU1079-001 1 mg 50.00 NU1079-005 5 mg 65.00 NU1079-010 10 mg 75.00 NU1079-050 50 mg 240.00 BMS387032 CDK2, CDK7, Serine-Threonine 345627-90-9 NU1080-001 1 mg 65.00 (SNS-032) CDK5, CDK4 NU1080-005 5 mg 110.00 NU1080-010 10 mg 175.00 NU1080-050 50 mg 605.00 TAK-715 p38 Serine-Threonine 303162-79-0 NU1087-001 1 mg 70.00 NU1087-005 5 mg 110.00 NU1087-010 10 mg 140.00 NU1087-050 50 mg 460.00 VX-702 P38 Serine-Threonine 745833-23-2 NU1093-001 1 mg 50.00 NU1093-005 5 mg 60.00 NU1093-010 10 mg 70.00 NU1093-050 50 mg 220.00 PHA690509 CDK2, CDK4, Serine-Threonine 492445-28-0 NU1097-001 1 mg 185.00 CDK5, CDK7 NU1097-005 5 mg 430.00 NU1097-010 10 mg 715.00 NU1097-050 50 mg 2,145.00 R1487 p38 Serine-Threonine 449808-64-4 NU1101-001 1 mg 180.00 (SY-R1487) NU1101-005 5 mg 385.00 NU1101-010 10 mg 605.00 NU1101-050 50 mg 1,815.00 VX745 MAPK Serine-Threonine 209410-46-8 NU1123-001 1 mg 80.00 NU1123-005 5 mg 130.00 NU1123-010 10 mg 190.00 NU1123-050 50 mg 620.00 BS194 CDK2, CDK1, CDK5, Serine-Threonine 1092443-55-4 NU1151-001 1 mg 195.00 CDK7, DK9 NU1151-005 5 mg 495.00 NU1151-010 10 mg 715.00 NU1151-050 50 mg 2,145.00 JNJ-28312141 GSK3, HER Serine-Threonine 885692-52-4 NU1154-001 1 mg 190.00 NU1154-005 5 mg 385.00 NU1154-010 10 mg 605.00 NU1154-050 50 mg 2,035.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 4
Lipid Kinase AS-252424 PI3K Lipid 900515-16-4 NU1009-001 1 mg 65.00 NU1009-005 5 mg 95.00 NU1009-010 10 mg 175.00 NU1009-050 50 mg 605.00 GDC-0941 PI3K Lipid 957054-30-7 NU1041-001 1 mg 80.00 (GDC0941) NU1041-005 5 mg 115.00 NU1041-010 10 mg 170.00 NU1041-050 50 mg 370.00 IC87114 PI3K Lipid 371242-69-2 NU1045-001 1 mg 60.00 NU1045-005 5 mg 90.00 NU1045-010 10 mg 160.00 NU1045-050 50 mg 550.00 PI103 PI3K, AKT, mtor Lipid 371935-74-9 NU1065-001 1 mg 95.00 NU1065-005 5 mg 145.00 NU1065-010 10 mg 230.00 NU1065-050 50 mg 450.00 PIK-93 PI3K Lipid 593960-11-3 NU1066-001 1 mg 105.00 NU1066-005 5 mg 170.00 NU1066-010 10 mg 260.00 NU1066-050 50 mg 1,045.00 PIK-75 PI3K Lipid 372196-67-3 NU1067-001 1 mg 50.00 NU1067-005 5 mg 65.00 NU1067-010 10 mg 75.00 NU1067-050 50 mg 275.00 PIK-90 PI3K Lipid 677338-12-4 NU1068-001 1 mg 50.00 NU1068-005 5 mg 70.00 NU1068-010 10 mg 120.00 NU1068-050 50 mg 355.00 TGX221 PI3K Lipid 663619-89-4 NU1089-001 1 mg 65.00 NU1089-005 5 mg 105.00 NU1089-010 10 mg 175.00 NU1089-050 50 mg 540.00 YM201636 PIKfyve Lipid 371942-69-7 NU1094-001 1 mg 100.00 NU1094-005 5 mg 160.00 NU1094-010 10 mg 250.00 NU1094-050 50 mg 850.00 PIK-294 PI3K Lipid 900185-02-6 NU1098-001 1 mg 105.00 NU1098-005 5 mg 160.00 NU1098-010 10 mg 290.00 NU1098-050 50 mg 890.00 ZSTK474 PI3K Lipid 475110-96-4 NU1099-001 1 mg 50.00 NU1099-005 5 mg 65.00 NU1099-010 10 mg 70.00 NU1099-050 50 mg 265.00 TG100115 PI3K Lipid 677297-51-7 NU1105-001 1 mg 100.00 NU1105-005 5 mg 165.00 NU1105-010 10 mg 265.00 NU1105-050 50 mg 760.00 LY294002 PI3K Lipid 154447-36-6 NU1108-001 1 mg 50.00 NU1108-005 5 mg 75.00 NU1108-010 10 mg 145.00 NU1108-050 50 mg 275.00 GNE-490 PI3K Lipid 1033739-92-2 NU1114-001 1 mg 190.00 NU1114-005 5 mg 385.00 NU1114-010 10 mg 540.00 NU1114-050 50 mg 1,375.00 GNE-493 PI3K Lipid 1033735-94-2 NU1115-001 1 mg 190.00 NU1115-005 5 mg 385.00 NU1115-010 10 mg 540.00 NU1115-050 50 mg 1,375.00 GSK2126458 PI3K Lipid 1086062-66-9 NU1126-001 1 mg 145.00 (HYR-582) NU1126-005 5 mg 220.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 5
GSK2126458 PI3K Lipid 1086062-66-9 NU1126-010 10 mg 350.00 (HYR-582) NU1126-050 50 mg 1,050.00 XL147 PI3K Lipid 956958-53-5 NU1127-001 1 mg 80.00 (SAR245408) NU1127-005 5 mg 130.00 NU1127-010 10 mg 160.00 NU1127-050 50 mg 450.00 XL765 PI3K Lipid 1349796-36-6 NU1137-001 1 mg 125.00 (SAR245409) NU1137-005 5 mg 210.00 NU1137-010 10 mg 320.00 NU1137-050 50 mg 1,045.00 NIBR-17 PI3K Lipid 944396-88-7 NU1145-001 1 mg 170.00 NU1145-005 5 mg 210.00 NU1145-010 10 mg 365.00 NU1145-050 50 mg 970.00 CH5132799 PI3K, mtor Lipid 1007207-67-1 NU1146-001 1 mg 125.00 NU1146-005 5 mg 210.00 NU1146-010 10 mg 320.00 NU1146-050 50 mg 950.00 GNE 477 PI3K Lipid 1032754-81-6 NU1148-001 1 mg 195.00 NU1148-005 5 mg 385.00 NU1148-010 10 mg 540.00 NU1148-050 50 mg 1,375.00 RG7422 PI3K Lipid 1032754-93-0 NU1150-001 1 mg 100.00 (GDC0980) NU1150-005 5 mg 150.00 NU1150-010 10 mg 250.00 NU1150-050 50 mg 750.00 BGT-226 PI3K Lipid 1245537-68-1 NU1178-001 1 mg 90.00 NU1178-005 5 mg 120.00 NU1178-010 10 mg 320.00 NU1178-050 50 mg 950.00 BGT-226 free base PI3K Lipid 915020-55-2 NU1178A-001 1 mg 90.00 NU1178A-005 5 mg 120.00 NU1178A-010 10 mg 320.00 NU1178A-050 50 mg 950.00 XL019 PI3K, mtor Lipid 945750-13-0 NU1191-001 1 mg 190.00 NU1191-005 5 mg 290.00 NU1191-010 10 mg 495.00 NU1191-050 50 mg 1,485.00 PF-04979064 PI3K, mtor Lipid 1220699-06-8 NU1194-001 1 mg 195.00 NU1194-005 5 mg 385.00 NU1194-010 10 mg 605.00 NU1194-050 50 mg 2,035.00 BKM120 PI3K, mtor Lipid 1312445-63-8 NU1200-001 1 mg 60.00 NU1200-005 5 mg 90.00 NU1200-010 10 mg 120.00 NU1200-050 50 mg 390.00 GDC-0032 PI3K Lipid 1282512-48-4 NU1202-001 1 mg 80.00 (GDC0032) NU1202-005 5 mg 120.00 NU1202-010 10 mg 200.00 NU1202-050 50 mg 650.00 PPI ABT-737 Bcl-2 852808-04-9 NU1001-001 1 mg 60.00 NU1001-005 5 mg 90.00 NU1001-010 10 mg 140.00 NU1001-050 50 mg 530.00 PTK AZ-960 JAK2 Tyrosine 905586-69-8 NU1015-001 1 mg 135.00 NU1015-005 5 mg 340.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 6
AZ-960 JAK2 Tyrosine 905586-69-8 NU1015-010 10 mg 540.00 NU1015-050 50 mg 1,300.00 Bosutinib Src, Abl Tyrosine 380843-75-4 NU1025-001 1 mg 50.00 (SKI-606) NU1025-005 5 mg 60.00 NU1025-010 10 mg 70.00 NU1025-050 50 mg 270.00 Tofacitinib JAK2 Tyrosine 477600-75-2 NU1032-001 1 mg 50.00 (CP690550, Xeljanz) NU1032-005 5 mg 70.00 NU1032-010 10 mg 90.00 NU1032-050 50 mg 240.00 Momelotinib JAK2 Tyrosine 1056634-68-4 NU1035-001 1 mg 80.00 (CYT387) NU1035-005 5 mg 110.00 NU1035-010 10 mg 160.00 NU1035-050 50 mg 450.00 Dasatinib Abl, BCR, BTK Tyrosine 302962-49-8 NU1036-001 1 mg 50.00 (BMS-354825, Sprycel) NU1036-005 5 mg 65.00 NU1036-010 10 mg 90.00 NU1036-050 50 mg 200.00 Dianilinopyrimidine_01 Pan Kinase Tyrosine 916603-07-1 NU1037-001 1 mg 150.00 NU1037-005 5 mg 350.00 NU1037-010 10 mg 500.00 NU1037-050 50 mg 1,050.00 Imatinib mesylate Abl, BCR Tyrosine 220127-57-1 NU1046-001 1 mg 40.00 (CGP54148, ST1571, NU1046-005 5 mg 55.00 Gleevec, Glivec) NU1046-010 10 mg 65.00 NU1046-050 50 mg 110.00 Merck 5 JAK Tyrosine 457081-03-7 NU1054-001 1 mg 195.00 NU1054-005 5 mg 485.00 NU1054-010 10 mg 695.00 NU1054-050 50 mg 1,980.00 PD173955 Abl, BCR Tyrosine 260415-63-2 NU1061-001 1 mg 165.00 NU1061-005 5 mg 275.00 NU1061-010 10 mg 430.00 NU1061-050 50 mg 1,375.00 PD173955-Analog1 Abl, BCR Tyrosine 185039-99-0 NU1062-001 1 mg 150.00 NU1062-005 5 mg 350.00 NU1062-010 10 mg 550.00 NU1062-050 50 mg 1,750.00 PF431396 PYK2 Tyrosine 717906-29-1 NU1063-001 1 mg 70.00 NU1063-005 5 mg 120.00 NU1063-010 10 mg 210.00 NU1063-050 50 mg 760.00 TG101209 JAK2 Tyrosine 936091-14-4 NU1103-001 1 mg 115.00 NU1103-005 5 mg 180.00 NU1103-010 10 mg 290.00 NU1103-050 50 mg 890.00 TG101348 JAK Tyrosine 936091-26-8 NU1104-001 1 mg 60.00 (SAR-302503) NU1104-005 5 mg 90.00 NU1104-010 10 mg 150.00 NU1104-050 50 mg 480.00 TG-46 JAK Tyrosine 936091-15-5 NU1106-001 1 mg 190.00 NU1106-005 5 mg 385.00 NU1106-010 10 mg 605.00 NU1106-050 50 mg 1,815.00 TG-89 JAK2 Tyrosine 936091-56-4 NU1107-001 1 mg 190.00 NU1107-005 5 mg 385.00 NU1107-010 10 mg 605.00 NU1107-050 50 mg 1,815.00 Mubritinib HER2 Tyrosine 366017-09-6 NU1112-001 1 mg 50.00 (TAK-165) NU1112-005 5 mg 65.00 NU1112-010 10 mg 70.00 NU1112-050 50 mg 275.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 7
Ponatinib Abl, BCR, FGFR Tyrosine 943319-70-8 NU1116-001 1 mg 60.00 (AP24534) NU1116-005 5 mg 90.00 NU1116-010 10 mg 110.00 NU1116-050 50 mg 365.00 Baricitinib JAK Tyrosine 1187595-84-1 NU1117-001 1 mg 165.00 (LY3009104, INCB-28050) NU1117-005 5 mg 275.00 NU1117-010 10 mg 385.00 NU1117-050 50 mg 1,155.00 Ruxolitinib JAK Tyrosine 941678-49-5 NU1120-001 1 mg 80.00 (INCB018424) NU1120-005 5 mg 140.00 NU1120-010 10 mg 200.00 NU1120-050 50 mg 600.00 R406 Syk Tyrosine 841290-80-0 NU1121-001 1 mg 100.00 NU1121-005 5 mg 165.00 NU1121-010 10 mg 250.00 NU1121-050 50 mg 850.00 Tamatinib fosdium BCR Tyrosine 1025687-58-4 NU1122-001 1 mg 105.00 (Fostamatinib, FosD, R788) NU1122-005 5 mg 165.00 NU1122-010 10 mg 300.00 NU1122-050 50 mg 970.00 RO495 TYK2 Tyrosine 1258296-60-4 NU1128-001 1 mg 195.00 NU1128-005 5 mg 485.00 NU1128-010 10 mg 695.00 NU1128-050 50 mg 1,980.00 NVP-BSK805 JAK2 Tyrosine 1092499-93-8 NU1136-001 1 mg 165.00 NU1136-005 5 mg 250.00 NU1136-010 10 mg 350.00 NU1136-050 50 mg 950.00 CEP-33779 JAK Tyrosine 1346168-57-7 NU1156-001 1 mg 145.00 NU1156-005 5 mg 240.00 NU1156-010 10 mg 385.00 NU1156-050 50 mg 1,265.00 GPLG0634 JAK1, JAK2 Tyrosine 1206161-97-8 NU1158-001 1 mg 190.00 NU1158-005 5 mg 320.00 NU1158-010 10 mg 460.00 NU1158-050 50 mg 1,310.00 PF4618433 PYK2, FAK Tyrosine 1166393-85-6 NU1163-001 1 mg 190.00 (PF-4618433) NU1163-005 5 mg 385.00 NU1163-010 10 mg 605.00 NU1163-050 50 mg 2,145.00 GCI1746 BTK Tyrosine 910232-84-7 NU1164-001 1 mg 165.00 (G-182) NU1164-005 5 mg 275.00 NU1164-010 10 mg 430.00 NU1164-050 50 mg 1,375.00 Ibrutinib BTK Tyrosine 936563-96-1 NU1171-001 1 mg 105.00 (PCI-32765) NU1171-005 5 mg 165.00 NU1171-010 10 mg 305.00 NU1171-050 50 mg 970.00 Bafetinib BCR Tyrosine 859212-16-1 NU1179-001 1 mg 100.00 (NS-187, INNO-406) NU1179-005 5 mg 170.00 NU1179-010 10 mg 310.00 NU1179-050 50 mg 940.00 Palbociclib HCl Abl, CDK2, CDK4, Tyrosine 827022-32-2 NU1180-001 1 mg 60.00 (PD-0332991) CDK5, CDK7 NU1180-005 5 mg 100.00 NU1180-010 10 mg 140.00 NU1180-050 50 mg 360.00 Palbociclib Isethionate Abl, CDK2, CDK4, Tyrosine 827022-33-3 NU1180A-001 1 mg 60.00 (PD-0332991) CDK5, CDK7 NU1180A-005 5 mg 100.00 NU1180A-010 10 mg 140.00 NU1180A-050 50 mg 360.00 RN486 BTK Tyrosine 1242156-23-5 NU1184-001 1 mg 350.00 NU1184-005 5 mg 950.00 NU1184-010 10 mg 1,450.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 8
CH4987655 MEK Tyrosine 874101-00-5 NU1188-001 1 mg 190.00 NU1188-005 5 mg 495.00 NU1188-010 10 mg 715.00 NU1188-050 50 mg 2,035.00 LY2784544 JAK2 Tyrosine 1229236-86-5 NU1196-001 1 mg 90.00 NU1196-005 5 mg 160.00 NU1196-010 10 mg 250.00 NU1196-050 50 mg 890.00 BLZ-945 c-fms Tyrosine 953769-46-5 NU1197-001 1 mg 160.00 NU1197-005 5 mg 350.00 NU1197-010 10 mg 550.00 NU1197-050 50 mg 1,850.00 GDC-046 TYK2 Tyrosine 1258292-64-6 NU1198-001 1 mg 90.00 (GDC046) NU1198-005 5 mg 150.00 NU1198-010 10 mg 240.00 NU1198-050 50 mg 850.00 PRT-060318 Syk Tyrosine 1194961-19-7 NU1204-001 1 mg 150.00 NU1204-005 5 mg 350.00 NU1204-010 10 mg 550.00 NU1204-050 50 mg 1,650.00 RTK Linifanib PDGFR Tyrosine 796967-16-3 NU1002-001 1 mg 80.00 (ABT-869, AL-39324, NU1002-005 5 mg 120.00 RG3635) NU1002-010 10 mg 200.00 NU1002-050 50 mg 550.00 Quizartinib PDGFR Tyrosine 950769-58-1 NU1003-001 1 mg 90.00 (AC220) NU1003-005 5 mg 190.00 NU1003-010 10 mg 310.00 NU1003-050 50 mg 890.00 AG13958 VEGF Tyrosine 319460-94-1 NU1004-001 1 mg 250.00 NU1004-005 5 mg 495.00 NU1004-010 10 mg 760.00 NU1004-050 50 mg 1,590.00 AMG-Tie2-1 Tie-2 Tyrosine 870223-96-4 NU1008-001 1 mg 195.00 NU1008-005 5 mg 390.00 NU1008-010 10 mg 590.00 NU1008-050 50 mg 1,815.00 AV-412 EGFR Tyrosine 451492-95-8 NU1012-001 1 mg 190.00 (MP-412) NU1012-005 5 mg 385.00 NU1012-010 10 mg 605.00 NU1012-050 50 mg 1,750.00 Tivozanib VEGFR Tyrosine 475108-18-0 NU1013-001 1 mg 80.00 (AV-951) NU1013-005 5 mg 130.00 NU1013-010 10 mg 185.00 NU1013-050 50 mg 605.00 Axitinib PDGFR Tyrosine 319460-85-0 NU1014-001 1 mg 45.00 (AG013736) NU1014-005 5 mg 55.00 NU1014-010 10 mg 65.00 NU1014-050 50 mg 70.00 BMS-2 MET Tyrosine 888719-03-7 NU1022-001 1 mg 250.00 NU1022-005 5 mg 750.00 NU1022-010 10 mg 1,250.00 CHIR-258 FGFR Tyrosine 405169-16-6 NU1029-001 1 mg 70.00 (TKI258) NU1029-005 5 mg 100.00 NU1029-010 10 mg 150.00 NU1029-050 50 mg 450.00 Canertinib EGFR Tyrosine 267243-28-7 NU1030-001 1 mg 50.00 (CI-1033, PD-183805) NU1030-005 5 mg 65.00 NU1030-010 10 mg 70.00 NU1030-050 50 mg 260.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 9
CP-724714 HER2 Tyrosine 383432-38-0 NU1033-001 1 mg 80.00 NU1033-005 5 mg 130.00 NU1033-010 10 mg 220.00 NU1033-050 50 mg 715.00 E7080 FGFR, VEGFR, SCF Tyrosine 417716-92-8 NU1038-001 1 mg 90.00 NU1038-005 5 mg 140.00 NU1038-010 10 mg 220.00 NU1038-050 50 mg 740.00 Erlotinib EGFR Tyrosine 183319-69-9 NU1039-001 1 mg 50.00 (OSI774, CP-358774, NU1039-005 5 mg 70.00 Tarceva, NSC718781) NU1039-010 10 mg 90.00 NU1039-050 50 mg 120.00 Gefitinib EGFR, HER2 Tyrosine 184475-35-2 NU1042-001 1 mg 40.00 (ZD1839, Iressa) NU1042-005 5 mg 55.00 NU1042-010 10 mg 65.00 NU1042-050 50 mg 120.00 GW441756 TrkA Tyrosine 504433-23-2 NU1044-001 1 mg 60.00 NU1044-005 5 mg 100.00 NU1044-010 10 mg 115.00 NU1044-050 50 mg 455.00 JNJ38877605 c-met Tyrosine 943540-75-8 NU1047-001 1 mg 90.00 NU1047-005 5 mg 130.00 NU1047-010 10 mg 210.00 NU1047-050 50 mg 750.00 Ki20227 c-fms Tyrosine 623142-96-1 NU1049-001 1 mg 100.00 NU1049-005 5 mg 165.00 NU1049-010 10 mg 240.00 NU1049-050 50 mg 825.00 Lapatinib EGFR Tyrosine 231277-92-2 NU1052-001 1 mg 50.00 (GW-572016, Tykerb) NU1052-005 5 mg 60.00 NU1052-010 10 mg 70.00 NU1052-050 50 mg 190.00 Masatinib c-kit, PDGFR, Tyrosine 790299-79-5 NU1053-001 1 mg 45.00 (AB1010, Masivet) FGFR3 NU1053-005 5 mg 60.00 NU1053-010 10 mg 90.00 NU1053-050 50 mg 350.00 Motesanib PDGFR Tyrosine 453562-69-1 NU1055-001 1 mg 65.00 (AMG706) NU1055-005 5 mg 110.00 NU1055-010 10 mg 175.00 NU1055-050 50 mg 550.00 Amuvatinib PDGFR Tyrosine 850879-09-3 NU1056-001 1 mg 100.00 (MP-470) NU1056-005 5 mg 190.00 NU1056-010 10 mg 315.00 NU1056-050 50 mg 850.00 Pazopanib PDGFR Tyrosine 444731-52-6 NU1058-001 1 mg 50.00 (GW786034, Votrient) NU1058-005 5 mg 60.00 NU1058-010 10 mg 70.00 NU1058-050 50 mg 150.00 Pazopanib HCl PDGFR Tyrosine 635702-64-6 NU1058A-001 1 mg 50.00 (GW786034, Votrient, NU1058A-005 5 mg 60.00 Armala) NU1058A-010 10 mg 70.00 NU1058A-050 50 mg 150.00 PF04217903 MET Tyrosine 956905-27-4 NU1060-001 1 mg 60.00 NU1060-005 5 mg 110.00 NU1060-010 10 mg 160.00 NU1060-050 50 mg 450.00 PF-562271 FGFR Tyrosine 717907-75-0 NU1064-001 1 mg 80.00 (PF562271) NU1064-005 5 mg 150.00 NU1064-010 10 mg 220.00 NU1064-050 50 mg 650.00 SB-216763 HER2 Tyrosine 280744-09-4 NU1075-001 1 mg 80.00 NU1075-005 5 mg 140.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 10
SB-216763 HER2 Tyrosine 280744-09-4 NU1075-010 10 mg 240.00 NU1075-050 50 mg 800.00 SU-5402 FGFR, PDGFR Tyrosine 215543-92-3 NU1084-001 1 mg 100.00 NU1084-005 5 mg 165.00 NU1084-010 10 mg 275.00 NU1084-050 50 mg 825.00 SU-6668 FGFR, PDGFR Tyrosine 252916-29-3 NU1085-001 1 mg 50.00 NU1085-005 5 mg 80.00 NU1085-010 10 mg 115.00 NU1085-050 50 mg 455.00 Sunitinib VEGFR2 (Flk-1), Tyrosine 341031-54-7 NU1086-001 1 mg 50.00 (SU11248) PDGFR NU1086-005 5 mg 75.00 NU1086-010 10 mg 100.00 NU1086-050 50 mg 145.00 Tandutinib PDGFR Tyrosine 387867-13-2 NU1088-001 1 mg 50.00 (CT53518, MLN518) NU1088-005 5 mg 65.00 NU1088-010 10 mg 75.00 NU1088-050 50 mg 90.00 Vandetanib EGFR, HER2 Tyrosine 443913-73-3 NU1090-001 1 mg 60.00 (ZD6474, Zactima) NU1090-005 5 mg 80.00 NU1090-010 10 mg 100.00 NU1090-050 50 mg 250.00 Intedanib FGFR, PDGFR Tyrosine 656247-17-5 NU1091-001 1 mg 80.00 (BIBF 1120, Vargatef ) NU1091-005 5 mg 120.00 NU1091-010 10 mg 190.00 NU1091-050 50 mg 650.00 KU57788 EGFR, HER2 Tyrosine 503468-95-9 NU1096-001 1 mg 50.00 (NU7441) NU1096-005 5 mg 75.00 NU1096-010 10 mg 110.00 Afatinib EGFR, HER2 Tyrosine 439081-18-2 NU1100-001 1 mg 80.00 (Tovok, BIBW-2992) NU1100-005 5 mg 120.00 NU1100-010 10 mg 200.00 NU1100-050 50 mg 550.00 AMG-25 PDGFR Tyrosine 1003311-62-3 NU1125-001 1 mg 190.00 NU1125-005 5 mg 495.00 NU1125-010 10 mg 760.00 NU1125-050 50 mg 2,200.00 Foretinib VEGFR2, MET Tyrosine 849217-64-7 NU1129-001 1 mg 105.00 (GSK1363089, EXEL-2880) NU1129-005 5 mg 160.00 NU1129-010 10 mg 290.00 NU1129-050 50 mg 850.00 Bayer-18 TYK2 Tyrosine 1251752-12-1 NU1130-001 1 mg 190.00 NU1130-005 5 mg 485.00 NU1130-010 10 mg 695.00 NU1130-050 50 mg 1,980.00 JNJ-38158471 VEGFR-2 Tyrosine 951151-97-6 NU1133-001 1 mg 190.00 NU1133-005 5 mg 385.00 NU1133-010 10 mg 540.00 NU1133-050 50 mg 1,485.00 BMS-540215 FGFR Tyrosine 649735-46-6 NU1134-001 1 mg 100.00 NU1134-005 5 mg 150.00 NU1134-010 10 mg 290.00 NU1134-050 50 mg 940.00 Brivanib FGFR Tyrosine 649735-63-7 NU1135-001 1 mg 145.00 (BMS-582664) NU1135-005 5 mg 240.00 NU1135-010 10 mg 350.00 NU1135-050 50 mg 900.00 Cabozantinib PDGFR Tyrosine 849217-68-1 NU1138-001 1 mg 65.00 (XL184, BMS-907351) NU1138-005 5 mg 110.00 NU1138-010 10 mg 170.00 NU1138-050 50 mg 460.00 Neratinib EGFR Tyrosine 698387-09-6 NU1140-001 1 mg 80.00 (HKI-272) NU1140-005 5 mg 120.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 11
Neratinib EGFR Tyrosine 698387-09-6 NU1140-010 10 mg 210.00 (HKI-272) NU1140-050 50 mg 715.00 Pelitinib EGFR, HER2 Tyrosine 257933-82-7 NU1141-001 1 mg 80.00 (EKB-569) NU1141-005 5 mg 120.00 NU1141-010 10 mg 210.00 NU1141-050 50 mg 715.00 BMS-599626 EGFR, HER2 Tyrosine 714971-09-2 NU1142-001 1 mg 105.00 (AC-480) NU1142-005 5 mg 165.00 NU1142-010 10 mg 275.00 NU1142-050 50 mg 870.00 AMG-1 c-met, RON Tyrosine 913376-84-8 NU1143-001 1 mg 165.00 NU1143-005 5 mg 275.00 NU1143-010 10 mg 430.00 NU1143-050 50 mg 1,530.00 Bentamapimod PDGFR Tyrosine 848344-36-5 NU1147-001 1 mg 190.00 (AS-602801) NU1147-005 5 mg 320.00 NU1147-010 10 mg 460.00 NU1147-050 50 mg 1,485.00 MK-2461 FGFR Tyrosine 917879-39-1 NU1149-001 1 mg 165.00 NU1149-005 5 mg 260.00 NU1149-010 10 mg 420.00 NU1149-050 50 mg 1,580.00 NVP-BGJ398 FGFR Tyrosine 872511-34-7 NU1152-001 1 mg 60.00 NU1152-005 5 mg 105.00 NU1152-010 10 mg 165.00 NU1152-050 50 mg 385.00 TAK-285 EGFR, HER2 Tyrosine 871026-44-7 NU1153-001 1 mg 165.00 NU1153-005 5 mg 260.00 NU1153-010 10 mg 455.00 NU1153-050 50 mg 1,620.00 SGX523 c-met Tyrosine 1072116-01-8 NU1155-001 1 mg 100.00 NU1155-005 5 mg 165.00 NU1155-010 10 mg 275.00 NU1155-050 50 mg 825.00 TAE684 ALK Tyrosine 761439-42-3 NU1159-001 1 mg 90.00 (NVP-TAE684) NU1159-005 5 mg 160.00 NU1159-010 10 mg 250.00 NU1159-050 50 mg 740.00 SAR131675 VEGFR-3 Tyrosine 1092539-44-0 NU1165-001 1 mg 190.00 NU1165-005 5 mg 385.00 NU1165-010 10 mg 605.00 NU1165-050 50 mg 2,145.00 Regorafenib VEGFR Tyrosine 835621-08-4 NU1169-001 1 mg 80.00 (BAY 73-4506) NU1169-005 5 mg 130.00 NU1169-010 10 mg 200.00 NU1169-050 50 mg 650.00 PD-0173074 VEGFR2, FGFR1 Tyrosine 219580-11-7 NU1176-001 1 mg 50.00 NU1176-005 5 mg 70.00 NU1176-010 10 mg 100.00 NU1176-050 50 mg 390.00 GNF-5837 TRK Serine-Threonine 1033769-28-6 NU1183-001 1 mg 80.00 NU1183-005 5 mg 130.00 NU1183-010 10 mg 200.00 NU1183-050 50 mg 715.00 SAR020106 EGFR, HER2 Tyrosine 1184843-57-9 NU1189-001 1 mg 190.00 NU1189-005 5 mg 385.00 NU1189-010 10 mg 605.00 NU1189-050 50 mg 1,860.00 LDK378 ALK Tyrosine 1032900-25-6 NU1199-001 1 mg 60.00 NU1199-005 5 mg 90.00 NU1199-010 10 mg 120.00 NU1199-050 50 mg 390.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 12
KW-2449 Aurora A, Abl, Tyrosine 841259-17-4 NU1205-001 1 mg 50.00 (KW2449) FGFR, BCR, fms NU1205-005 5 mg 70.00 NU1205-010 10 mg 90.00 NU1205-050 50 mg 270.00 RTK, PTK Nilotinib Abl, PDGFR, BCR Tyrosine 641571-10-0 NU1057-001 1 mg 50.00 (AMN107, Tasigna) NU1057-005 5 mg 70.00 NU1057-010 10 mg 100.00 NU1057-050 50 mg 150.00 STE CI-1040 MEK, MKK4&7, MKK3&6, Serine-Threonine 212631-79-3 NU1031-001 1 mg 50.00 (PD184352) MEK5, MEK2, MEK1 NU1031-005 5 mg 70.00 NU1031-010 10 mg 120.00 NU1031-050 50 mg 430.00 PD0325901 MEK Serine-Threonine 391210-10-9 NU1059-001 1 mg 50.00 NU1059-005 5 mg 70.00 NU1059-010 10 mg 120.00 NU1059-050 50 mg 430.00 S-99 ASK Serine-Threonine 1124381-69-6 NU1119-001 1 mg 190.00 NU1119-005 5 mg 385.00 NU1119-010 10 mg 605.00 NU1119-050 50 mg 2,035.00 Crizotinib MEK1, MEK2, MKK3&6, Serine-Threonine 877399-52-5 NU1139-001 1 mg 60.00 (PF-02341066) MKK4&7, MEK, MEK5 NU1139-005 5 mg 110.00 NU1139-010 10 mg 165.00 NU1139-050 50 mg 560.00 MLN0128 MEK, MEK5, Serine-Threonine 1224844-38-5 NU1157-001 1 mg 95.00 (INK-128) MEK2, MEK1 NU1157-005 5 mg 160.00 NU1157-010 10 mg 260.00 NU1157-050 50 mg 930.00 GSK1120212 MEK1, MEK2 Serine-Threonine 871700-17-3 NU1170-001 1 mg 80.00 (JTP-74057, GSK212, NU1170-005 5 mg 115.00 Trametinib) NU1170-010 10 mg 205.00 NU1170-050 50 mg 645.00 PP242 MEK, MEK5, Serine-Threonine 1092351-67-1 NU1181-001 1 mg 50.00 MEK2, MEK1 NU1181-005 5 mg 70.00 NU1181-010 10 mg 110.00 NU1181-050 50 mg 365.00 CX6258 PKC, PKCalpha Serine-Threonine 1202916-90-2 NU1182-001 1 mg 190.00 NU1182-005 5 mg 320.00 NU1182-010 10 mg 460.00 NU1182-050 50 mg 1,375.00 MPI0479605 MEK, MEK5 Serine-Threonine 1246529-32-7 NU1187-001 1 mg 190.00 NU1187-005 5 mg 320.00 NU1187-010 10 mg 495.00 NU1187-050 50 mg 1,485.00 AS703026 MEK1, MEK2 Serine-Threonine 1236699-92-5 NU1190-001 1 mg 60.00 NU1190-005 5 mg 90.00 NU1190-010 10 mg 120.00 NU1190-050 50 mg 390.00 ARRY 334543 MEK, MEK2, Serine-Threonine 845272-21-1 NU1192-001 1 mg 90.00 (ARRY 33454 ) MEK5, MEK1 NU1192-005 5 mg 190.00 NU1192-010 10 mg 290.00 NU1192-050 50 mg 990.00 AZD8330 MEK1, MEK2 Serine-Threonine 869357-68-6 NU1195-001 1 mg 100.00 NU1195-005 5 mg 170.00 NU1195-010 10 mg 320.00 NU1195-050 50 mg 940.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 13
TKL AMG-47a LIMK Serine-Threonine 882663-88-9 NU1007-001 1 mg 195.00 NU1007-005 5 mg 385.00 NU1007-010 10 mg 610.00 NU1007-050 50 mg 1,750.00 BMS-3 LIMK1, LIMK2 Serine-Threonine 1338247-30-5 NU1023-001 1 mg 190.00 NU1023-005 5 mg 385.00 NU1023-010 10 mg 605.00 NU1023-050 50 mg 1,815.00 BMS-5 LIMK1, LIMK2 Serine-Threonine 1338247-35-0 NU1024-001 1 mg 190.00 NU1024-005 5 mg 385.00 NU1024-010 10 mg 605.00 NU1024-050 50 mg 1,815.00 PLX4720 ARaf, Raf, CRaf, BRaf Tyrosine 918505-84-7 NU1069-001 1 mg 60.00 NU1069-005 5 mg 90.00 NU1069-010 10 mg 115.00 NU1069-050 50 mg 385.00 SB590885 ARaf, Raf, CRaf, BRaf Serine-Threonine 405554-55-4 NU1077-001 1 mg 80.00 NU1077-005 5 mg 130.00 NU1077-010 10 mg 170.00 NU1077-050 50 mg 655.00 Sorafenib ARaf, CRaf, BRaf Serine-Threonine 284461-73-0 NU1082-001 1 mg 50.00 (Nexavar, BAY43-9006) NU1082-005 5 mg 65.00 NU1082-010 10 mg 75.00 NU1082-050 50 mg 275.00 PLX4032 Raf Serine-Threonine 918504-65-1 NU1161-001 1 mg 50.00 (Vemurafenib, RG7204, NU1161-005 5 mg 65.00 Zelboraf, RO5185426) NU1161-010 10 mg 75.00 NU1161-050 50 mg 260.00 Takeda-6d B-RAF, VEGFR2 Serine-Threonine 1125632-93-0 NU1168-001 1 mg 195.00 NU1168-005 5 mg 385.00 NU1168-010 10 mg 605.00 NU1168-050 50 mg 1,815.00 TAK632 Raf Serine-Threonine 1228591-30-7 NU1203-001 1 mg 70.00 NU1203-005 5 mg 120.00 NU1203-010 10 mg 170.00 NU1203-050 50 mg 650.00 Other AT9283 Aurora A Serine-Threonine 896466-04-9 NU1011-001 1 mg 80.00 NU1011-005 5 mg 150.00 NU1011-010 10 mg 250.00 NU1011-050 50 mg 740.00 (R)-BI-2536 Plk1 Serine-Threonine 755038-02-9 NU1019-001 1 mg 80.00 NU1019-005 5 mg 115.00 NU1019-010 10 mg 195.00 NU1019-050 50 mg 650.00 CYC116 Aurora A Serine-Threonine 693228-63-6 NU1034-001 1 mg 60.00 NU1034-005 5 mg 90.00 NU1034-010 10 mg 120.00 NU1034-050 50 mg 350.00 JNJ-7706621 Aurora A, CDK7, CDK5, Serine-Threonine 443797-96-4 NU1048-001 1 mg 125.00 CDK4, CDK2 NU1048-005 5 mg 210.00 NU1048-010 10 mg 355.00 NU1048-050 50 mg 835.00 SNS-314 Aurora A Serine-Threonine 1057249-41-8 NU1081-001 1 mg 80.00 NU1081-005 5 mg 130.00 NU1081-010 10 mg 200.00 NU1081-050 50 mg 650.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 14
Tozasertib Aurora A Serine-Threonine 639089-54-6 NU1092-001 1 mg 50.00 (MK-0457, VX-680) NU1092-005 5 mg 65.00 NU1092-010 10 mg 75.00 NU1092-050 50 mg 220.00 Danusertib Abl, Aurora A, Serine-Threonine 827318-97-8 NU1095-001 1 mg 105.00 (PHA-739358) BCR, FGFR NU1095-005 5 mg 170.00 NU1095-010 10 mg 310.00 NU1095-050 50 mg 950.00 GSK2606414 PERK Serine-Threonine 1337531-89-1 NU1201-001 1 mg 90.00 NU1201-005 5 mg 160.00 NU1201-010 10 mg 250.00 NU1201-050 50 mg 690.00 PF-05274857 hydrochloride Smo 1373615-35-0 NU3008-001 1 mg 145.00 (PF05274857 hydrochloride) NU3008-005 5 mg 250.00 NU3008-010 10 mg 430.00 NU3008-050 50 mg 1,590.00 Epigenetics (+)-JQ1 BET bromodomain 1268524-70-4 NU3004-001 1 mg 125.00 NU3004-005 5 mg 210.00 NU3004-010 10 mg 365.00 NU3004-050 50 mg 1,045.00 PF-06405761 BRD4 1403764-72-6 NU3009-001 1 mg 90.00 (PF06405761) NU3009-005 5 mg 140.00 NU3009-010 10 mg 155.00 NU3009-050 50 mg 450.00 GPCR ER 172594-06 474550-69-1 NU3002-001 1 mg 195.00 (Atopaxar hydrobromide, NU3002-005 5 mg 460.00 E5555) NU3002-010 10 mg 715.00 NU3002-050 50 mg 2,145.00 Pfizer Licensed PF-04981517 CYP3A4, CYP3A4, 1390637-82-7 NU3007-001 1 mg 50.00 (CYP3CIDE) CYP3A5, CYP3A7 NU3007-005 5 mg 90.00 NU3007-010 10 mg 190.00 NU3007-050 50 mg 600.00 Azithromycin Bacterial Ribosime (50S) 83905-01-5 NU3010-001 1 mg 50.00 (Zithromax, Azithrocin, NU3010-005 5 mg 65.00 Azin) NU3010-010 10 mg 75.00 NU3010-050 50 mg 165.00 Torcetrapib CETP 262352-17-0 NU3011-001 1 mg 60.00 (CP-529414) NU3011-005 5 mg 100.00 NU3011-010 10 mg 165.00 NU3011-050 50 mg 570.00 Voriconazole 137234-62-9 NU3012-001 1 mg 50.00 (VFEND-UK-109-496) NU3012-005 5 mg 60.00 NU3012-010 10 mg 70.00 NU3012-050 50 mg 275.00 Varenicline tartrate Nicotinic ACh 375815-87-5 NU3013-001 1 mg 60.00 (Chantix, Champix) receptor (a4b2) NU3013-005 5 mg 90.00 NU3013-010 10 mg 170.00 NU3013-050 50 mg 540.00 UK-383367 BMP-1 348622-88-8 NU3014-001 1 mg 50.00 NU3014-005 5 mg 65.00 NU3014-010 10 mg 75.00 NU3014-050 50 mg 275.00 Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 15
Celecoxib COX-2 169590-42-5 NU3015-001 1 mg 50.00 (Geodon) NU3015-005 5 mg 55.00 NU3015-010 10 mg 60.00 NU3015-050 50 mg 65.00 Sildenafil Citrate PDE5 171599-83-0 NU3016-001 1 mg 50.00 (Viagra, Revatio) NU3016-005 5 mg 110.00 NU3016-010 10 mg 200.00 NU3016-050 50 mg 275.00 Prazosin hydrochloride Alpha-1 receptors, 19237-84-4 NU3017-001 1 mg 50.00 (Minipress, Vasoflex, MT3 receptor NU3017-005 5 mg 65.00 Pressin) NU3017-010 10 mg 75.00 NU3017-050 50 mg 275.00 Sulbactam beta-lactamase 68373-14-8 NU3018-001 1 mg 50.00 NU3018-005 5 mg 65.00 NU3018-010 10 mg 75.00 NU3018-050 50 mg 275.00 Ziprasidone hydrochloride 138982-67-9 NU3019-001 1 mg 50.00 hydrate NU3019-005 5 mg 65.00 (Geodon) NU3019-010 10 mg 75.00 NU3019-050 50 mg 275.00 Atorvastatin calcium HMG-CoA reductase 134523-03-8 NU3020-001 1 mg 50.00 (Lipitor) NU3020-005 5 mg 65.00 NU3020-010 10 mg 75.00 NU3020-050 50 mg 110.00 Linezolid Ribosome (23S) 165800-03-3 NU3021-001 1 mg 50.00 (Zyvox) NU3021-005 5 mg 65.00 NU3021-010 10 mg 75.00 NU3021-050 50 mg 275.00 Nelfinavir Mesylate 159989-65-8 NU3022-001 1 mg 50.00 (AG 1341) NU3022-005 5 mg 65.00 NU3022-010 10 mg 75.00 NU3022-050 50 mg 275.00 Exemestane Aromatase 107868-30-4 NU3023-001 1 mg 50.00 (FCE 24304) NU3023-005 5 mg 65.00 NU3023-010 10 mg 70.00 NU3023-050 50 mg 260.00 Tigecycline Bacterial Ribosime (30S) 220620-09-7 NU3024-001 1 mg 60.00 (GAR 936, Glycylcycline, NU3024-005 5 mg 90.00 Tygacil, WAY-GAR 936) NU3024-010 10 mg 110.00 NU3024-050 50 mg 385.00 Alprostadil 745-65-3 NU3025-001 1 mg 80.00 (Caverject, Prostaglandin E1) NU3025-005 5 mg 120.00 NU3025-010 10 mg 155.00 NU3025-050 50 mg 495.00 Glyburide SUR1 10238-21-8 NU3026-001 1 mg 50.00 (Diabeta, Glibenclamide) NU3026-005 5 mg 65.00 NU3026-010 10 mg 75.00 NU3026-050 50 mg 100.00 Miglitol 72432-03-2 NU3027-001 1 mg 60.00 (Glyset) NU3027-005 5 mg 90.00 NU3027-010 10 mg 110.00 NU3027-050 50 mg 385.00 Adalat 1829-25-4 NU3028-001 1 mg 50.00 (Cordipin, Nifedical, Procardia, NU3028-005 5 mg 65.00 BAY 1040, Nifediac) NU3028-010 10 mg 75.00 NU3028-050 50 mg 100.00 Storage: 4C Nacalai USA, Inc. 10225 Barnes Canyon Rd., Suite A 103, San Diego, CA 92121 info@nacalaiusa.com www.nacalaiusa.com Page 16